![icon logo Griffin Discoveries](http://www.griffindiscoveries.com/wp-content/themes/Griffin/images/icon_logo.jpg)
![rat H1R binding](http://www.griffindiscoveries.com/images/rat H1R binding.png)
Type of assay | Biochemical |
Receptor: | Rat Histamine H1 |
Expression system: | Transient transfection of HEK-293T |
Radioligand: | [3H]mepyramine |
Radioligand concentration: | 1.3 nM |
Kd (nM): | 1 nM |
Experiment settings: | - 8 concentrations of test compounds, each in triplicate – total reaction volume of 200 µL – incubation at RT for 1 hour |
Read-out: | Scintillation counting, converted in dpm unit |
Reference: | Cetirizine (Ki = 8 nM) |
Z’ factor | >0.7 |